MCHR1 antagonist 3

• UNSPSC Description:

  MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism[1].

• Target Antigen:

  MCHR1 (GPR24)

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;Neuronal Signaling

• Applications:

  Metabolism-protein/nucleotide metabolism

• Field of Research:

  Endocrinology; Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/mchr1-antagonist-3.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(N1C2CC3=C(C=CC=C3)C2)N(CC)C4(CCN(CC5=CC=C(N6CCCC6)C=C5)CC4)C1=O

• Molecular Weight:

  472.62

• References & Citations:

  [1]Rowbottom MW, et al. Synthesis and structure-activity relationships of spirohydantoin-derived small-moleculeantagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Bioorg Med Chem Lett. 2007 Apr 15;17(8):2171-8.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  1069622-60-1