Products for Research Use Only
RegisterLogin

TGR5 agonist 5

CAT: 0804-HY-161817Size: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-161817Size:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
TGR5 agonist 5 (compound K91) is a potent agonist of TGR5, with EC50s of 19 μM and 30 μM in CRE-Luciferase assay anf cAMP accumulation assay, respectively[1].
UNSPSC
12352005
Target
G protein-coupled Bile Acid Receptor 1
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/tgr5-agonist-5.html
Smiles
CC1(C)N(CC(NC[C@H]2OC3=CC=CC=C3C2)=O)CCC4=CC=CC=C41
Molecular Formula
C22H26N2O2
Molecular Weight
350.45
References & Citations
[1]M Giovanna E Papadopoulos, et al. Discovery and characterization of small-molecule TGR5 ligands with agonistic activity. Eur J Med Chem. 2024 Jun 28:276:116616.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-149807TGR5 agonist 1
HY-14229-01TGR5 Receptor Agonist
HY-155306TGR5 agonist 3
HY-168140TGR5 agonist 6
HY-149808TGR5 agonist 2
HY-168329TGR5 agonist 7
HY-155307TGR5 agonist 4
HY-146453TGR5 Receptor Agonist 3
HY-156830-01TGR5 Receptor Agonist 4
HY-142159FXR/TGR5 agonist 1

Alternative Products

CatalogName
B1185-5TGR5 Receptor Agonist
T203565-01TGR5 agonist 7
T200705-01TGR5 agonist 6
SD2384-5mgTGR5 (GPCR19 agonist)
GTR19220890-01TGR5 agonist 1
GTR19218689-01TGR5 agonist 3
GTR19274766-01TGR5 agonist 9
T74825-01TGR5 agonist 2
B1635-25TGR5-Receptor-Agonist
GTR19231323-01TGR5 agonist 4

Popular Products