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CP-809101

CAT: 0804-HY-15543Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-15543Size:1 Each
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Description
CP-809101 is a potent and highly selective 5-HT2C receptor agonist, with pEC50s of 9.96, 7.19 and 6.81 M for human 5HT2C, 5HT2B and 5HT2A receptor. CP-809101 inhibits conditioned avoidance responding in rats and antagonizes both PCP (phencyclidine hydrochloride) - and d-amphetamine-induced hyperactivity. CP-809101 also reduces food and nicotine dependence in rats, can be used in studies of antipsychotic and nicotine dependence[1][2].
CAS Number
479683-64-2
UNSPSC
12352005
Hazard Statement
H315-H319-H320
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cp-809101.html
Solubility
10 mM in DMSO
Smiles
ClC1=CC(COC2=NC(N3CCNCC3)=CN=C2)=CC=C1
Molecular Formula
C15H17ClN4O
Molecular Weight
304.77
Precautions
P264-P280-P302+P352-P305+P351+P338-P362
References & Citations
[1]Siuciak JA, et al. CP-809,101, a selective 5-HT2C agonist, shows activity in animal models of antipsychotic activity. Neuropharmacology. 2007 Feb;52 (2) :279-90. |[2]Higgins GA, et al. Evaluation of chemically diverse 5-HT₂c receptor agonists on behaviours motivated by food and nicotine and on side effect profiles. Psychopharmacology (Berl) . 2013 Apr;226 (3) :475-90.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor; α-1 microglobulin

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