PF-CBP1
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


PF-CBP1
UNSPSC Description:
PF-CBP1 is a highly selective inhibitor of the CREB binding protein bromodomain[1].Target Antigen:
Epigenetic Reader DomainType:
Reference compoundRelated Pathways:
EpigeneticsApplications:
Neuroscience-NeurodegenerationField of Research:
Neurological DiseaseAssay Protocol:
https://www.medchemexpress.com/pf-cbp1.htmlSolubility:
10 mM in DMSOSmiles:
CCCOC1=CC=C(CCC2=NC3=CC(C4=C(C)ON=C4C)=CC=C3N2CCN5CCOCC5)C=C1Molecular Weight:
488.62References & Citations:
[1]Chekler EL, et al. Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. Chem Biol. 2015 Dec 17;22(12):1588-96.Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
1962928-21-7
