PF-04781340
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


PF-04781340
UNSPSC Description:
PF-04781340 is a potent and selective 5-HT2C receptor agonist. PF-04781340 is orally available and have central nervous system penetrant profile[1].Target Antigen:
5-HT ReceptorType:
Reference compoundRelated Pathways:
GPCR/G Protein;Neuronal SignalingApplications:
Neuroscience-NeuromodulationField of Research:
Neurological DiseaseAssay Protocol:
https://www.medchemexpress.com/pf-04781340.htmlSolubility:
10 mM in DMSOSmiles:
CNC1=NC(CC2=CC=CC=C2)=CC3=C1CCNCC3Molecular Weight:
267.37References & Citations:
[1]Rouquet G, et al. Design, Synthesis, and Evaluation of Tetrasubstituted Pyridines as Potent 5-HT2C Receptor Agonists. ACS Med Chem Lett. 2015 Jan 20;6(3):329-33.Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
1648726-56-0
