DPI-287

• UNSPSC Description:

  DPI-287 is a selective delta-opioid receptor (DOP) agonist with a Ki value of 0.39 nM and can be used for pain research[1].

• Target Antigen:

  Opioid Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;Neuronal Signaling

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/dpi-287.html

• Solubility:

  10 mM in DMSO

• Smiles:

  C[C@@H](CN([C@@H](C1)C)CC2=CC=CC=C2)N1[C@@H](C3=CC(O)=CC=C3)C4=CC=C(C=C4)C(N(CC)CC)=O

• Molecular Weight:

  485.66

• References & Citations:

  [1]Claff T, et al. Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists. Sci Adv. 2019 Nov 27;5(11):eaax9115.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  519058-13-0