DPI-287

• Description:

  DPI-287 is a selective delta-opioid receptor (DOP) agonist with a Ki value of 0.39 nM and can be used for pain research[1].

• UNSPSC:

  12352005

• Target:

  Opioid Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/dpi-287.html

• Solubility:

  10 mM in DMSO

• Smiles:

  C[C@@H] (CN ([C@@H] (C1) C) CC2=CC=CC=C2) N1[C@@H] (C3=CC (O) =CC=C3) C4=CC=C (C=C4) C (N (CC) CC) =O

• Molecular Formula:

  C31H39N3O2

• Molecular Weight:

  485.66

• References & Citations:

  [1]Claff T, et al. Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists. Sci Adv. 2019 Nov 27;5 (11) :eaax9115.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  519058-13-0