DPI-287

• Description :

  DPI-287 is a selective delta-opioid receptor (DOP) agonist with a Ki value of 0.39 nM and can be used for pain research[1].

• UNSPSC :

  12352005

• Target :

  Opioid Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Neuronal Signaling

• Applications :

  Neuroscience-Neuromodulation

• Field of Research :

  Neurological Disease

• Assay Protocol :

  https://www.medchemexpress.com/dpi-287.html

• Solubility :

  10 mM in DMSO

• Smiles :

  C[C@@H](CN([C@@H](C1)C)CC2=CC=CC=C2)N1[C@@H](C3=CC(O)=CC=C3)C4=CC=C(C=C4)C(N(CC)CC)=O

• Molecular Formula :

  C31H39N3O2

• Molecular Weight :

  485.66

• References & Citations :

  [1]Claff T, et al. Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists. Sci Adv. 2019 Nov 27;5 (11) :eaax9115.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• CAS Number :

  [519058-13-0]