PSB-1901

• UNSPSC Description:

  PSB-1901 is a potent A2B adenosine receptor (A2BAR) antagonist with Kis of 0.0835 nM and 0.131 nM for human and mouse A2BARs respectively. PSB-1901 can be used for the research of cancer[1].

• Target Antigen:

  Adenosine Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/psb-1901.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C1NC2=C(C(N1CCC)=O)NC(C3=CC=C(S(=O)(N4CCN(CC4)C5=CC=C(C=C5)Br)=O)C=C3)=N2

• Molecular Weight:

  573.46

• References & Citations:

  [1]Jiang J, et al. A2B Adenosine Receptor Antagonists with Picomolar Potency. J Med Chem. 2019 Apr 25;62(8):4032-4055.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  2332835-02-4