BRD7-IN-3

CAT: 0804-HY-149421Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-149421Size:1 Each
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Description
BRD7-IN-3 (compound 1-78) is a dual inhibitor of bromodomain-containing proteins BRD7/BRD9 with IC50s of 1.6 μM and 2.7 μM respectively[1].
CAS Number
[3032601-04-7]
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/brd7-in-3.html
Solubility
10 mM in DMSO
Smiles
CC1=CC(N(C2=C1C=CC(C3=CC=C(N=C3C)OC)=C2)C)=O
Molecular Formula
C18H18N2O2
Molecular Weight
294.35
References & Citations
[1]Ordonez-Rubiano SC, et al. Rational Design and Development of Selective BRD7 Bromodomain Inhibitors and Their Activity in Prostate Cancer. J Med Chem. 2023 Aug 24;66 (16) :11250-11270..
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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