BRD7-IN-2

• Target:

  Epigenetic Reader Domain

• Related Pathways:

  Chromatin/Epigenetic

• Bioactivity:

  BRD7-IN-2 (compound 2-77) is a potent, selective inhibitor of bromodomain-containing protein 7 (BRD7) with an IC50 of 5.4 ?M and exhibits significant anti-proliferative activity in prostate cancer cells, while demonstrating weak inhibition of BRD9 with an IC50 of >300 ?M.

• Molecular Formula:

  C18H18N2O3

• Molecular Weight:

  310.35

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C