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GPR81 agonist 2

CAT: 0804-HY-148563Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-148563Size:1 Each
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Description
GPR81 agonist 2 (compound 1) is a potent GPR81 agonist with EC50 values of 0.023, 0.123 µM for hGPR81, hGPR109A, respectively[1].
CAS Number
1143024-28-5
UNSPSC
12352005
Target
Hydroxycarboxylic Acid Receptor (HCAR)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/gpr81-agonist-2.html
Solubility
10 mM in DMSO
Smiles
O=C(NC1=NC2=C(S1)C=C(S(=O)(C3CCN(CC3)C)=O)C=C2)NC(C4=C(Cl)C=C(OCC)C(N5N=CC=C5)=C4)=O
Molecular Formula
C26H27ClN6O5S2
Molecular Weight
603.11
References & Citations
[1]Davidsson Ö, et al. Identification of novel GPR81 agonist lead series for target biology evaluation. Bioorg Med Chem Lett. 2020 Feb 15;30 (4) :126953.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
HCAR1

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