DC-CPin7

• Description :

  DC-CPin7 is a potent inhibitor of CREB-binding protein (CBP) bromodomain with an IC50 of 2.5 μM[1].

• UNSPSC :

  12352005

• Target :

  Epigenetic Reader Domain

• Type :

  Reference compound

• Related Pathways :

  Epigenetics

• Applications :

  Cancer-programmed cell death

• Field of Research :

  Cancer

• Assay Protocol :

  https://www.medchemexpress.com/dc-cpin7.html

• Solubility :

  10 mM in DMSO

• Smiles :

  OC(C1C(CC=CC1)C(NC2=CC3=C(C=C2)N(C(OC)=O)CCC3)=O)=O

• Molecular Formula :

  C19H22N2O5

• Molecular Weight :

  358.39

• References & Citations :

  [1]Chen Y, et al. Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain. Bioorg Chem. 2020 Aug;101:103991.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• CAS Number :

  [893781-17-4]