GPCR modulator-1

• Description:

  GPCR modulator-1 is a negative allosteric modulator of GLP receptor. GPCR modulator-1 has the potential for type 2 diabetes research[1].

• UNSPSC:

  12352005

• Target:

  GCGR

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  Metabolism-sugar/lipid metabolism

• Field of Research:

  Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/gpcr-modulator-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(O)CCNC(C1=CC=C([C@@H](C2CC(C)(C)C2)NC3=CC=C(N4C=C(C(F)(F)F)N=C4)N=C3)C=C1)=O

• Molecular Formula:

  C26H28F3N5O3

• Molecular Weight:

  515.53

• References & Citations:

  [1]Gaojie Song, et al. Human GLP-1 receptor transmembrane domain structure in complex with allosteric modulators. Nature. 2017 Jun 8;546 (7657) :312-315.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  [1407592-99-7]