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CB1 inverse agonist 2

CAT: 0804-HY-12095-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-12095-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CB1 inverse agonist 2 is an orally active inverse agonist of Cannabinoid Receptor CB1. CB1 inverse agonist 2 effectively inhibits CP55940-induced hypothermia and anorexia in mice model[1].
CAS Number
1019839-52-1
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cb1-inverse-agonist-2.html
Purity
99.15
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC=C2SC3=CC=CC=C3C(C4=CC=C(F)C(Cl)=C4)=NC2=C1)NCCCC
Molecular Formula
C24H20ClFN2OS
Molecular Weight
438.94
References & Citations
[1]Synthesis and Evaluation of Dibenzothiazepines: A Novel Class of Selective Cannabinoid-1 Receptor Inverse Agonists J. Med. Chem., 2009, 52 (7), pp 1975-1982|[2]Pettersson H, et al. Synthesis and evaluation of dibenzothiazepines: a novel class of selective cannabinoid-1 receptor inverse agonists. J Med Chem. 2009 Apr 9;52 (7) :1975-82.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, stored under nitrogen)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB1; CB2

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