CB1/2 agonist 2

• Description:

  CB1/2 agonist 2 (compound 23) is a potent non-selective cannabinoid ligand, with Ki values of 3.5 and 1.2 nM, respectively. CB1/2 agonist 2 can behave as a full CB1 agonist and CB2 competitive inverse agonist. CB1/2 agonist 2 shows antinociceptive activity[1].

• UNSPSC:

  12352005

• Target:

  Cannabinoid Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling

• Applications:

  COVID-19-immunoregulation

• Field of Research:

  Inflammation/Immunology

• Assay Protocol:

  https://www.medchemexpress.com/cb1-2-agonist-2.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(NC1CC1)CCCCCCCCCCOC2=CC(CCCCC)=CC(OC)=C2

• Molecular Formula:

  C26H43NO3

• Molecular Weight:

  417.62

• References & Citations:

  [1]Brizzi A, et al. Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity. Bioorg Med Chem. 2020 Jun 1;28 (11) :115513.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• Isoform:

  CB1; CB2

• CAS Number:

  [2772379-97-0]