RegisterLogin

PQ-69

CAT: 0804-HY-110186Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-110186Size:1 Each
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
PQ-69 is a potent and selective adenosine A1 receptor antagonist with inverse agonist activity. PQ-69 binds to hA1 receptor with a Ki value of 0.96 nM, is 217-fold more selective compared with hA2A receptors (Ki=208 nM) and >1,000-fold selectivity over hA3 receptor (Ki >100 μM) . PQ-69 can be used for the research of renal dysfunction[1].
CAS Number
[910045-32-8]
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/pq-69.html
Solubility
10 mM in DMSO
Smiles
O=C1N(C2=CC=CC(F)=C2)NC3=C1C(NCCCC)=NC4=CC=CC=C34
Molecular Formula
C20H19FN4O
Molecular Weight
350.39
References & Citations
[1]Min Lu, et al. PQ-69, a novel and selective adenosine A1 receptor antagonist with inverse agonist activity. Purinergic Signal. 2014 Dec;10 (4) :619-29.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-18078-01PQ-10
HY-14584PQ-1
HY-14584APQ-1 (succinate)
HY-161229HSD17B13-IN-69
HY-139892XR8-69
HY-162697α-Glucosidase-IN-69
HY-114402-01ARD-69
HY-159116AChE-IN-69
HY-124022HDAC-IN-69
HY-170836NLRP3-IN-69

Alternative Products

CatalogName
T28446-01PQ-69
T24656-01PQ-10
2768/50PQ 401
564631PQ-912
A11951-25PQ 401 25mg
A11951-50PQ 401 50mg

Popular Products