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PD-217014

CAT: 0804-HY-136644ASize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-136644ASize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PD-217014 is an α2δ ligand with visceral analgesic activity and can inhibit visceral hypersensitivity reactions. Its anti-allodynic effect is dose-dependent.
CAS Number
335458-65-6
UNSPSC
12352211
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/pd-217014.html
Smiles
OC(C[C@@]1(C[C@@]2([H])[C@@](CC2)([H])C1)CN)=O
Molecular Formula
C10H17NO2
Molecular Weight
183.25
References & Citations
[1]Effect of a new alpha 2 delta ligand PD-217014 on visceral hypersensitivity induced by 2,4,6-trinitrobenzene sulfonic acid in rats
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported