RUPB-61

CAT: 0804-HY-161309Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-161309Size:1 Each
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
RUPB-61 is a potent Plasmodium falciparum cGMP-dependent protein kinase (PfPKG) inhibitor with an IC50 value of 13 nM. RUPB-61 shows antiparasitic activity[1].
UNSPSC
12352005
Target
Parasite
Type
Reference compound
Related Pathways
Anti-infection
Applications
COVID-19-immunoregulation
Field of Research
Infection
Assay Protocol
https://www.medchemexpress.com/pfpkg-in-2.html
Solubility
10 mM in DMSO
Smiles
FC(C=C1)=CC=C1C(NC([C@@H]2[C@H](C)CN(C)CC2)=C3)=C3C4=CC=NC=C4
Molecular Formula
C22H24FN3
Molecular Weight
349.44
References & Citations
[1]Gilleran JA, et al. Structure-Activity Relationship of a Pyrrole Based Series of PfPKG Inhibitors as Anti-Malarials. J Med Chem. 2024 Feb 19.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-114956AT-61
HY-163258HSD17B13-IN-61
HY-121769BFE-61
HY-179160Tubulin-IN-61
HY-176733HDAC6-IN-61
HY-13901-01GANT 61
HY-147860EGFR-IN-61
HY-P2428RI-61
HY-100025HLCL-61
HY-163825RNB-61

Alternative Products

CatalogName
MBS5779821AT 61
MBS3604680-01GANT 61
T89580-01RNB-61
T73128-01EGFR-IN-61
T86651-01HSD17B13-IN-61
MBS5812091Mpro 61
526868HT-61
B7806-25HLCL-61
BA3015-1ARD-61
T204999-01RNB 61

Popular Products