BRD4-IN-9

BRD4-IN-9

• CAS Number: 2468959-08-0
• UNSPSC Description: BRD4-IN-9 is an orally active BRD4 inhibitor with an IC50 value of 9.4 nM. BRD4-IN-9 can suppress tumor growth in a mouse melanoma xenograft model[1].
• Target Antigen: Others
• Type: Reference compound
• Related Pathways: Others
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/brd4-in-9.html
• Smiles: CN(C(C=C1)=O)C=C1C2=CC=C(N=C(C3CCOCC3)N4)C4=C2OC5=CC=CC=C5
• Molecular Weight: 401.46
• References & Citations: [1]Horai Y, et al. A novel 7-phenoxy-benzimidazole derivative as a potent and orally available BRD4 inhibitor for the treatment of melanoma. Bioorg Med Chem. 2024 Oct 1;112:117882.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported