BRD4-IN-4

CAT: 0804-HY-153751-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-153751-01Size:5 mg
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Description
BRD4-IN-4 (Compound 1) is a BRD4 inhibitor (IC50=6.83 μM) . BRD4-IN-4 selectively inhibits MV4-11 cell line proliferation and arrests cell at G1 phase. BRD4-IN-4 can be used for research of MLL leukemia[1].
CAS Number
[304685-40-3]
UNSPSC
12352005
Hazard Statement
H302-H315-H319
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/brd4-in-4.html
Purity
96.0
Solubility
DMSO : 100 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C1C2=CC=CC3=C(S(=O)(N4CCCC4)=O)C=CC(N1CC)=C32
Molecular Formula
C17H18N2O3S
Molecular Weight
330.40
Precautions
P264-P270-P280-P302+P352-P305+P351+P338-P330-P362+P364-P501
References & Citations
[1]Feng Y, et al. Design, synthesis and biological evaluation of benzo[cd]indol-2 (1H) -ones derivatives as BRD4 inhibitors. Eur J Med Chem. 2018 May 25;152:264-273.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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