LY 301875

• Description :

  LY 301875 is a potent and orally active angiotensin II receptor type 1 (AT1) antagonist with a pKB value of 9.6[1].

• UNSPSC :

  12352005

• Target :

  Angiotensin Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein

• Field of Research :

  Cardiovascular Disease

• Assay Protocol :

  https://www.medchemexpress.com/ly-301875.html

• Smiles :

  CCCCCC[C@@H](N1C=C(N=C1)NC(C2=C(C=CC=C2)S(=O)(O)=O)=O)C(N3[C@@H](C[C@@H](C3)OC4=CC=C(C=C4)CC(O)=O)C(O)=O)=O

• Molecular Formula :

  C31H36N4O10S

• Molecular Weight :

  656.70

• References & Citations :

  [1]Boyd, D. B., et al. Molecular Modeling and Quantitative Structure—Activity Relationship Studies in Pursuit of Highly Potent Substituted Octanoamide Angiotensin II Receptor Antagonists. Computer-Aided Molecular Design, 1995, 14-35.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• Isoform :

  AT1 Receptor

• CAS Number :

  [154668-27-6]