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UFP-512

CAT: 0804-HY-130176Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-130176Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
UFP-512 is a selective and potent σ-opioid receptor (DOP receptor) peptidic agonist with antidepressant- and anxiolytic-like effects. UFP-512 exhibits as a potent agonist on adenylyl cyclase inhibition and Erk1/2 activation. UFP-512 induces phosphorylation of DOP receptors on Ser363 with a low desensitization of the cAMP pathway. UFP-512 is promising for research of mood disorders[1].
CAS Number
480446-44-4
UNSPSC
12352005
Target
Adenylate Cyclase; ERK; Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; MAPK/ERK Pathway; Neuronal Signaling; Stem Cell/Wnt
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ufp-512.html
Smiles
CC(C=C(C=C1C)O)=C1C[C@H](N)C(N2[C@@H](CC3=CC=CC=C3C2)C(N[C@H](C4=NC5=CC=CC=C5N4)CC(O)=O)=O)=O
Molecular Formula
C31H33N5O5
Molecular Weight
555.62
References & Citations
[1]Aguila B, et al. In vitro and in vivo pharmacological profile of UFP-512, a novel selective delta-opioid receptor agonist; correlations between desensitization and tolerance. Br J Pharmacol. 2007 Dec;152 (8) :1312-24.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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