UFP-803

CAT: 0931-TP2104Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-TP2104Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
879497-82-2
Target
GPCR
Related Pathways
GPCR/G Protein|||Endocrinology/Hormones
Bioactivity
Urotensin-II (UT) receptor ligand; behaves as a silent antagonist in most in vitro assays and in vivo, but does retain small residual agonist activity under certain conditions in some assays. Competitively antagonizes U-II induced contractions in the rat aorta (pIC50 = 7.46) and prevents plasma extravasation elicited by U-II in mice in vivo.
Smiles
C(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@@H](NC([C@H](CC(O)=O)N)=O)C(C)(C)SSC[C@@H](C(N[C@@H](C(C)C)C(O)=O)=O)NC(=O)[C@H](CC5=CC=C(O)C=C5)NC(=O)[C@H](CCN)NC3=O
Molecular Formula
C50H64N10O12S2
Molecular Weight
1061.24
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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