PI3Kα Ligand-1

CAT: 0804-HY-174798Size: 1 EachDry Ice: NoHazardous: No

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CAT#:0804-HY-174798Size:1 Each

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Description

PI3Kα Ligand-1 is the ligand for PI3Kα that can be used for synthesis of PROTACs, such as PI3Kα degrader-1.

UNSPSC

12352005

Target

Ligands for Target Protein for PROTAC; PI3K

Related Pathways

PI3K/Akt/mTOR; PROTAC

Field of Research

Cancer

Smiles

O=S(NC1=C(N=CC(C2=CC3=C(N=CN=C3C(O)=C2)C)=C1)OC)(C4=CC=C(C=C4F)F)=O

Molecular Formula

C21H16F2N4O4S

Molecular Weight

458.44

References & Citations

[1]Peng S, et al. Discovery and Optimization of Potent PROTAC Degraders of Phosphoinositide 3-Kinase with Significant in Vivo Anticancer Efficacy. J Med Chem. 2025 Jun 26;68 (12) :12800-12818.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

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T1826-01	PI3K-IN-1
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PI3Kα Ligand-1

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