GRL-098-22

• Description :

  GRL-098-22 (Compound 6t) is a potent inhibitor targeting G protein-coupled receptor kinase 5 (GRK5) and GRK6 with IC50 values of 0.6 μM and 0.19 μM, respectively. GRL-098-22 is promising for research of diseases such as heart failure and multiple myeloma[1].

• UNSPSC :

  12352005

• Target :

  G Protein-coupled Receptor Kinase (GRK)

• Related Pathways :

  GPCR/G Protein

• Field of Research :

  Cancer; Cardiovascular Disease

• Smiles :

  O=C(N1C[C@@H](C(NC2=C(C)NC(/C=C3C(NC4=C\3C=C(C(N[C@@H](C5=CC=C(F)C=C5)C)=O)C=C4)=O)=C2C)=O)NCC1)OC(C)(C)C

• Molecular Formula :

  C34H39FN6O5

• Molecular Weight :

  630.71

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported