Products for Research Use Only

IRL-1038 TFA

CAT: 0931-TP2262L1-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-TP2262L1-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Endothelin Receptor
Related Pathways
GPCR/G Protein
Purity
0.9879
Bioactivity
IRL-1038 TFA is a selective and potent endothelin B (ETB) receptor antagonist that inhibits endothelin-induced endothelium-dependent relaxation and can be used in the study of cardiovascular disease.
Smiles
O=C([C@H]1NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CSSC1)N)=O)C(C)C)=O)CC2=CC=C(C=C2)O)=O)CC3=CC=CC=C3)=O)N[C@@H](CC4=CN=CN4)C(N[C@@H](CC(C)C)C(N[C@@H](CC(O)=O)C(N[C@@H]([C@@H](C)CC)C(N[C@@H]([C@@H](C)CC)C(N[C@H](C(O)=O)CC5=CNC6=CC=CC=C56)=O)=O)=O)=O)=O.OC(C(F)(F)F)=O
Molecular Formula
C70H93F3N14O17S2
Molecular Weight
1523.7
Shipping Conditions
Ice Packs
Storage Temperature
-20°C