IRL 2500

• Target:

  Endothelin Receptor

• Related Pathways:

  GPCR/G Protein

• Purity:

  0.9936

• Bioactivity:

  IRL 2500 is an antagonist of Endothelin receptor with IC50s of 1.3 and 94 nM for Endothelin A receptor and Endothelin B receptor.

• Smiles:

  CN([C@H](Cc1ccc(cc1)-c1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(O)=O)C(=O)c1cc(C)cc(C)c1

• Molecular Formula:

  C36H35N3O4

• Molecular Weight:

  573.68

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  169545-27-1