IRL-1620 acetate

• Target:

  Endothelin Receptor

• Related Pathways:

  GPCR/G Protein

• Purity:

  0.9664

• Bioactivity:

  IRL-1620 acetate is an effective and selective agonist of Endothelin B receptor (ETB) with a Ki of 16 pM which is more selective than ETA with a Ki of 19 ?M.

• Smiles:

  CC (O) =O.O=C (O) [C@H] (CC1=CNC2=C1C=CC=C2) NC ([C@H] ([C@@H] (C) CC) NC ([C@H] ([C@@H] (C) CC) NC ([C@H] (CC (O) =O) NC ([C@H] (CC (C) C) NC ([C@H] (CC3=CNC=N3) NC ([C@H] (C) NC ([C@H] (CC4=CC=CC=C4) NC ([C@H] (CC5=CC=C (O) C=C5) NC ([C@H] (C (C) C) NC ([C@H] (C) NC ([C@H] (CCC (O) =O) NC ([C@H] (CCC (O) =O) NC ([C@H] (CC (O) =O) NC (CCC (O) =O) =O) =O) =O) =O) =O) =O) =O) =O) =O) =O) =O) =O) =O) =O

• Molecular Formula:

  C88H121N17O29

• Molecular Weight:

  1881

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C