M4 mAChR Modulator-1

CAT: 0931-MF-0122081-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0122081-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
AChR
Related Pathways
Neuroscience
Bioactivity
M4 mAChR Modulator-1 (compound 23i) acts as a positive allosteric modulator (PAM) of the M4 mAChR. It demonstrates a stronger synergistic effect in ?-arrestin recruitment compared to G protein activation when interacting with ACh. Additionally, while its PAM effects are weaker in G protein-mediated responses, they are more potent in ?-arrestin recruitment.
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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