BChE-IN-20

• Target :

  Cholinesterase (ChE) |||Others

• Related Pathways :

  Neuroscience|||Others

• Bioactivity :

  BChE-IN-20 (compound 7c) is a potent and selective inhibitor of BChE, with IC50 values of 105 nM for eqBChE and 2.3 nM for hBChE. It also inhibits P glycoprotein with an IC50 of 0.27 ?M. BChE-IN-20 serves as a promising template for the design and development of pharmaceutical BChE-selective ligands, including inhibitors and fluorogenic probes.

• Smiles :

  O=C(OC)C1=CN(CCC=2N=C(N=C(NCCCN(CC)CC)C2C1)C=3C=CC=CC3)C(C)C

• Molecular Formula :

  C27H39N5O2

• Molecular Weight :

  465.63

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1428439-79-5