ABCG2-IN-2

• Target:

  BCRP

• Related Pathways:

  Membrane transporter/Ion channel

• Bioactivity:

  ABCG2-IN-2 is a potent inhibitor of ABCG2, showing favorable oral pharmacokinetic profiles in mice, and is applicable for investigating tumor multidrug resistance (MDR) and erythropoietic protoporphyria (EPP) [1].

• Smiles:

  C(C(C)C)[C@H]1C2=C(C=3C(N2)=CC(OC)=CC3)C[C@@]4(N1C(=O)[C@H](CCC(NC(C)C)=O)NC4=O)[H]

• Molecular Formula:

  C25H34N4O4

• Molecular Weight:

  454.56

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2559759-59-8