CARM1-IN-3

• Target :

  Histone Methyltransferase

• Related Pathways :

  Chromatin/Epigenetic

• Bioactivity :

  CARM1-IN-3 (compound 17b) is a potent and selective inhibitor of co-activator associated arginine methyltransferase (CARM1), with IC50 values of 0.07 µM for CARM1 and greater than 25 µM for CARM3 [1].

• Smiles :

  O(C)C1=C(C(OC)=CC=C1)C=2NC=3C(N2)=C(C)C=C(C3)C4CCN(CCNC)CC4

• Molecular Formula :

  C24H32N4O2

• Molecular Weight :

  408.54

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  912970-67-3