CARM1-IN-5
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


CARM1-IN-5
Target :
Histone MethyltransferaseRelated Pathways :
Chromatin/EpigeneticBioactivity :
CARM1-IN-5 (Compound 17e) is a potent and selective inhibitor of CARM1, exhibiting an IC50 of 2 nM. By directly interacting with CARM1, CARM1-IN-5 effectively inhibits the methylation of substrate proteins. Additionally, CARM1-IN-5 demonstrates significant antiproliferative effects on melanoma cell lines.Shipping Conditions :
Cool packStorage Temperature :
-20°C

