Products for Research Use Only

Elabela (19-32) TFA

CAT: 0931-T76044-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T76044-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Apelin receptor, Arrestin
Related Pathways
GPCR/G Protein
Bioactivity
Elabela (19-32) TFA, an effective fragment of ELABELA (ELA), selectively engages with the apelin receptor (APJ) . This compound initiates G αi1 and β-arrestin-2 signaling, demonstrating EC50 values of 8.6 nM and 166 nM, respectively. It facilitates receptor internalization, lowers arterial pressure, and has a positive inotropic impact on cardiac function [1].
Molecular Formula
C77H120F3N25O19S2
Molecular Weight
1821.05
Shipping Conditions
Ice Packs
Storage Temperature
-20°C