Products for Research Use Only

CTAP TFA

CAT: 0931-T75917-01Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T75917-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Target
Opioid Receptor
Related Pathways
Endocrinology/Hormones, GPCR/G Protein, Neuroscience
Bioactivity
CTAP TFA, a potent and highly selective μ opioid receptor antagonist that effectively crosses the blood-brain barrier, exhibits a significant inhibition concentration (IC50) of 3.5 nM. It demonstrates extraordinary selectivity, being over 1200-fold more specific to μ opioid receptors than to δ opioid (IC50 = 4500 nM) and somatostatin receptors. This compound is primarily leveraged for researching L-DOPA-induced dyskinesia (LID) and opiate overdose or addiction [1] [2].
Molecular Formula
C53H70F3N13O12S2
Molecular Weight
1218.32
Shipping Conditions
Ice Packs
Storage Temperature
-20°C