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CAT: 0931-TP2050Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-TP2050Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
103429-32-9
Target
Opioid Receptor
Related Pathways
Endocrinology/Hormones, GPCR/G Protein, Neuroscience
Bioactivity
Potent and selective μ opioid receptor antagonist (IC50 = 3.5 nM) . Displays > 1200-fold selectivity over δ opioid and somatostatin receptors. Brain penetrant and active in vivo.
Smiles
C[C@@H](O)[C@H](NC(=O)C1NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CSSC1(C)C)NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(N)=O
Molecular Formula
C51H69N13O11S2
Molecular Weight
1104.32
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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