CTAP

• Target:

  Opioid Receptor

• Related Pathways:

  Endocrinology/Hormones|||GPCR/G Protein|||Neuroscience

• Bioactivity:

  Potent and selective ? opioid receptor antagonist (IC50 = 3.5 nM) . Displays > 1200-fold selectivity over ? opioid and somatostatin receptors. Brain penetrant and active in vivo.

• Smiles:

  C[C@@H](O)[C@H](NC(=O)C1NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CSSC1(C)C)NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(N)=O

• Molecular Formula:

  C51H69N13O11S2

• Molecular Weight:

  1104.32

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  103429-32-9