CTAP

• Target :

  Opioid Receptor

• Related Pathways :

  Endocrinology/Hormones|||GPCR/G Protein|||Neuroscience

• Bioactivity :

  Potent and selective ? opioid receptor antagonist (IC50 = 3.5 nM) . Displays > 1200-fold selectivity over ? opioid and somatostatin receptors. Brain penetrant and active in vivo.

• Smiles :

  C[C@@H](O)[C@H](NC(=O)C1NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CSSC1(C)C)NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(N)=O

• Molecular Formula :

  C51H69N13O11S2

• Molecular Weight :

  1104.32

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  103429-32-9