TD-802

• Target :

  PROTACs|||Androgen Receptor|||Others

• Related Pathways :

  Others|||Endocrinology/Hormones|||PROTAC

• Bioactivity :

  TD-802 (Compound 33c), an androgen receptor (AR) PROTAC degrader, exhibits strong microsomal stability and demonstrates potent antitumor efficacy in vivo, making it suitable for research on metastatic castration-resistant prostate cancer [1].

• Smiles :

  CC1(C)[C@H](NC(=O)c2ccc(cc2)N2CCN(CC2)C2CC3(C2)CCN(CC3)C(=O)C2CCN(CC2)c2ccc3nnn(C4CCC(=O)NC4=O)c(=O)c3c2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1

• Molecular Formula :

  C52H61ClN10O6

• Molecular Weight :

  957.56

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2760703-21-5