Cyclo (RLsKDK)

• CAS Number :

  1975145-82-4

• Target :

  MMP

• Related Pathways :

  Proteases/Proteasome

• Bioactivity :

  Cyclo (RLsKDK) (BK-1361) serves as a targeted inhibitor of the metalloproteinase ADAM8, demonstrating efficacy with an IC50 value of 182 nM. This compound shows promise for use in the treatment of inflammatory diseases and cancer, highlighting its potential therapeutic applications.

• Smiles :

  C(CCNC(=N)N)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)[C@H](CC(C)C)NC1=O

• Molecular Formula :

  C31H57N11O9

• Molecular Weight :

  727.85

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C