PQM-244

• Target:

  Cannabinoid Receptor|||TRP/TRPV Channel

• Related Pathways:

  GPCR/G Protein|||Membrane transporter/Ion channel

• Bioactivity:

  PQM-244 (Compound 5c) is an orally active multi-target modulator that acts on TRPV1, CB1, and CB2 receptors. It exhibits significant peripheral analgesic effects during both neurogenic and inflammatory phases. PQM-244 also shows potential antioxidant activity with a DPPH radical scavenging IC50 of 14.15 µM. This compound is applicable for research into chronic pain and inflammatory diseases, such as diabetes, atherosclerosis, and Alzheimer's disease.

• Smiles:

  O=C(NN=C1C(=CCC(C(=C)C)C1)C)C2=CC=C(OC)C=C2

• Molecular Formula:

  C18H22N2O2

• Molecular Weight:

  298.38

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  316139-50-1