PQM-244

CAT: 0931-T211171-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-T211171-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
316139-50-1
Target
Cannabinoid Receptor|||TRP/TRPV Channel
Related Pathways
GPCR/G Protein|||Membrane transporter/Ion channel
Bioactivity
PQM-244 (Compound 5c) is an orally active multi-target modulator that acts on TRPV1, CB1, and CB2 receptors. It exhibits significant peripheral analgesic effects during both neurogenic and inflammatory phases. PQM-244 also shows potential antioxidant activity with a DPPH radical scavenging IC50 of 14.15 µM. This compound is applicable for research into chronic pain and inflammatory diseases, such as diabetes, atherosclerosis, and Alzheimer's disease.
Smiles
O=C(NN=C1C(=CCC(C(=C)C)C1)C)C2=CC=C(OC)C=C2
Molecular Formula
C18H22N2O2
Molecular Weight
298.38
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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