Products for Research Use Only

TRK-IN-31

CAT: 0931-T211064-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T211064-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Trk receptor
Related Pathways
Tyrosine Kinase/Adaptors
Bioactivity
TRK-IN-31 is an orally active TRK inhibitor with an IC50 of 1.8 nM. It demonstrates excellent antiproliferative activity in Ba/F3-MPRIP-TRKAG667C cells and selectively inhibits TRK kinase activity effectively. TRK-IN-31 also significantly suppresses tumor growth in a Ba/F3-MPRIP-TRKAG667C subcutaneous tumor mouse model.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C