α2AR agonist 1

• Target:

  Adrenergic Receptor

• Related Pathways:

  GPCR/G Protein|||Neuroscience

• Bioactivity:

  ?2AR agonist 1 (compound S6a) is a morpholinopyrimidinone that serves as an agonist for the ?2-adrenergic receptor (?2AR) . This compound elicits a concentration-dependent relaxation in precontracted aortic rings induced by phenylephrine (pEC50=6.81) . Additionally, ?2AR agonist 1 elevates levels of NOx and NO in HUVEC.

• Molecular Formula:

  C16H15N4NaO2

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C