α2AR agonist 2
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α2AR agonist 2
Description :
α2AR agonist 2 is a selective α2B adrenergic receptor antagonist (IC50 = 1.2 µM) . α2AR agonist 2 can be used for research on inflammatory pain and neuropathic pain[1].CAS Number :
[719277-27-7]UNSPSC :
12352005Target :
Adrenergic ReceptorRelated Pathways :
GPCR/G Protein; Neuronal SignalingField of Research :
Inflammation/Immunology; Neurological DiseaseSmiles :
CCN1C2=CC(F)=CC=C2S/C1=C\C(C)=OMolecular Formula :
C12H12FNOSMolecular Weight :
237.29References & Citations :
[1]Hagiwara, et al. Pharmaceutical composition containing alpha-2 adrenergic receptor antagonist for analgesia. WO2022065354 A1.Shipping Conditions :
Room temperatureScientific Category :
Reference compound1Clinical Information :
No Development Reported

