Products for Research Use Only

CI-988 hemihydrate

CAT: 0931-T208995-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T208995-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Cholecystokinin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
CI-988 hemihydrate (PD134308) is a potent and selective orally active CCK2R (cholecystokinin 2 receptor) antagonist, with an IC50 of 1.7 nM for mouse cortical CCK2. It is over 1600 times more selective for CCK2 than for CCK1 receptors. CI-988 hemihydrate exhibits anxiolytic and antitumor properties.
Molecular Formula
C35H42N4O6.1/2H2O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C