CB1R agonist 1

• Target:

  Cannabinoid Receptor

• Related Pathways:

  GPCR/G Protein

• Bioactivity:

  CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.

• Smiles:

  CC1=CC(C(N[C@@](C(OC)=O)(C)C2=CC=CS2)=O)=NN1C3=CC(C(F)(F)F)=CC=C3

• Molecular Formula:

  C20H18F3N3O3S

• Molecular Weight:

  437.435

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C