Gefapixant citrate

• Description:

  Gefapixant citrate is an orally active P2X3 receptor (P2X3R) antagonist that acts on human homologous recombinant hP2X3 (IC50: ~30 nM) and hP2X2/3 (IC50: 100-200 nM) . Gefapixant citrate can be used to study chronic cough and knee osteoarthritis.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  545.52

• Molecular Formula:

  C20H27N5O11S

• Notes:

  Research use only, not for human use.

• Receptor:

  Others

• CAS Number:

  2310299-91-1