Gefapixant

• Description:

  Gefapixant (AF-219, MK-7264) is an orally active, small molecule antagonist of P2X3-containing receptor with IC50 of 30 nM (hP2X3 homotrimer) and 100-250 nM (hP2X2/3 heterotrimer) .

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  353.397

• Molecular Formula:

  C14H19N5O4S

• Notes:

  Research use only, not for human use.

• Receptor:

  RecombinanthP2X3homotrimers|hP2X2/3heterotrimericreceptors

• CAS Number:

  1015787-98-0