Products for Research Use Only

Gefapixant

CAT: 1410-M10082-01Size: 1 EachDry Ice: NoHazardous: No
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CAT#:1410-M10082-01Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Gefapixant (AF-219, MK-7264) is an orally active, small molecule antagonist of P2X3-containing receptor with IC50 of 30 nM (hP2X3 homotrimer) and 100-250 nM (hP2X2/3 heterotrimer) .
CAS Number
1015787-98-0
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
353.397
Molecular Formula
C14H19N5O4S
Notes
Research use only, not for human use.
Receptor
RecombinanthP2X3homotrimers|hP2X2/3heterotrimericreceptors