PARP10-IN-2
CAT:
804-HY-148753-03
Size:
10 mg
Price:
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
PARP10-IN-2
- CAS Number: 1042780-52-8
- UNSPSC Description: PARP10-IN-2 is a potent mono‐ADP‐ribosyltransferase PARP10 inhibitor with an IC50 of 3.64 μM for human PARP10. PARP10-IN-2 reveals potent inhibition on PARP2 and PARP15 with IC50s of 27 μM and 11 μM for human PARP2 and human PARP15, respectively[1].
- Target Antigen: PARP
- Type: Reference compound
- Related Pathways: Cell Cycle/DNA Damage;Epigenetics
- Applications: Cancer-programmed cell death
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/parp10-in-2.html
- Solubility: DMSO : 250 mg/mL (ultrasonic)
- Smiles: N#CC1=CC=C(C=C1)OC2=CC=C(C(N)=O)C=C2
- Molecular Weight: 238.24
- References & Citations: [1]Patricia Korn, et al. Evaluation of 3- and 4-Phenoxybenzamides as Selective Inhibitors of the Mono-ADP-Ribosyltransferase PARP10. ChemistryOpen. 2021 Oct;10(10):939-948.
- Shipping Conditions: Blue Ice
- Clinical Information: No Development Reported