ARTD10/PARP10-IN-1
CAT:
804-HY-148709
Size:
Inquire
Price:
Ask
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
ARTD10/PARP10-IN-1
- CAS Number: 1708103-76-7
- UNSPSC Description: ARTD10/PARP10-IN-1 (compound 23) is a potent and non-selective PARP inhibitor, targeting to mono-ADP-ribosyltransferases ARTD7/PARP15, ARTD8/PARP14, ARTD10/PARP10 and poly(ADP-ribose) polymerase-1 (ARTD1/PARP1) with IC50s of 1.7 μM, 1.6 μM, 0.8 μM, and 4.4 μM, respectively[1].
- Target Antigen: PARP
- Type: Reference compound
- Related Pathways: Cell Cycle/DNA Damage;Epigenetics
- Applications: COVID-19-anti-virus
- Field of Research: Inflammation/Immunology
- Assay Protocol: https://www.medchemexpress.com/artd10-parp10-in-1.html
- Solubility: 10 mM in DMSO
- Smiles: COC(/C=C\C(NC1=CC(C(N)=O)=CC=C1)=O)=O
- Molecular Weight: 248.23
- References & Citations: [1]Ekblad T, et al. Towards small molecule inhibitors of mono-ADP-ribosyltransferases. Eur J Med Chem. 2015 May 5;95:546-51.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported