Products for Research Use Only

Nav1.8-IN-16

CAT: 0013-GTR19257949-01Size: 50 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0013-GTR19257949-01Size:50 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Nav1.8-IN-16 (Compound (R) -40) is an orally bioavailable and selective hNaV 1.8 inhibitor with an IC50 of 5.9 nM. It provides analgesic effects by blocking the NaV1.8 channel without significantly affecting other NaV subtypes or the hERG channel. Nav1.8-IN-16 demonstrates dose-dependent pain relief in postoperative and inflammatory pain models and is suitable for pain-related research.
Field of Research
Pharmacology & Drug Discovery
Molecular Formula
C24H16ClF5N2O3
Storage Conditions
-20°C
Notes
For research use only.