Products for Research Use Only

AR antagonist 9

CAT: 0013-GTR19241366-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19241366-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
AR antagonist 9 is a potent, orally bioavailable androgen receptor (AR) antagonist that disrupts AR dimerization. It exhibits activity comparable to Enzalutamide against wild-type AR and shows superior efficacy against common resistance mutants like ARF876L/T877A. This compound demonstrates significant oral bioavailability and inhibits tumor growth in LNCaP xenograft models, supporting its research in overcoming prostate cancer resistance.
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Molecular Formula
C18H13F4NO2
Molecular Weight
351.29
Storage Conditions
-20°C
Notes
For research use only.

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