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PROTAC BRM degrader-1

CAT: 0013-GTR19234726-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19234726-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PROTAC BRM degrader-1 (compound 17) is a potent, heterobifunctional degrader of the SWI/SNF ATPase subunits BRM (SMARCA2) and BRG1 (SMARCA4), with DC50 values of 93 pM and 4.9 nM, respectively. This tool compound enables the study of chromatin remodeling in cancer research, applicable for both in vitro and in vivo mechanistic investigations.
CAS Number
2378051-80-8
Field of Research
Epigenetics & Chromatin, Neuroscience, Pharmacology & Drug Discovery
Smiles
O (C1=CC (N2C3CN (CC2CC3) C=4C=C (N=NC4N) C5=C (O) C=CC=C5) =CC=N1) [C@@H]6C[C@@H] (OC7CCN (CCOC=8C=C ([C@H] (C (=O) N9[C@H] (C (N[C@@H] (C) C%10=CC=C (C=C%10) C=%11SC=NC%11C) =O) C[C@@H] (O) C9) C (C) C) ON8) CC7) C6
Molecular Formula
C57H69N11O8S
Molecular Weight
1068.29
Storage Conditions
-20°C
Notes
For research use only.

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